Vijender Panduga
Bellary Road
Bengaluru, KA 560024, India
Bengaluru, KA 560024, India
Last Updated: 09/26/2026
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Found 18 publications
Scaffold Morphing To Identify Novel DprE1 Inhibitors with Antimycobacterial Activity.
Journal: ACS medicinal chemistry letters
Published: July 29, 2019
Discovery of Imidazo[1,2-a]pyridine Ethers and Squaramides as Selective and Potent Inhibitors of Mycobacterial Adenosine Triphosphate (ATP) Synthesis.
Journal: Journal of medicinal chemistry
Published: January 12, 2017
Evaluation of the metabolism, bioactivation and pharmacokinetics of triaminopyrimidine analogs toward selection of a potential candidate for antimalarial therapy.
Journal: Xenobiotica; the fate of foreign compounds in biological systems
Published: October 19, 2016
In silico-based high-throughput screen for discovery of novel combinations for tuberculosis treatment.
Journal: Antimicrobial agents and chemotherapy
Published: December 26, 2014
Triaminopyrimidine is a fast-killing and long-acting antimalarial clinical candidate.
Journal: Nature communications
Published: September 15, 2014
N-aryl-2-aminobenzimidazoles: novel, efficacious, antimalarial lead compounds.
Journal: Journal of medicinal chemistry
Published: July 10, 2014
1,4-azaindole, a potential drug candidate for treatment of tuberculosis.
Journal: Antimicrobial agents and chemotherapy
Published: June 25, 2014
Aminoazabenzimidazoles, a novel class of orally active antimalarial agents.
Journal: Journal of medicinal chemistry
Published: June 11, 2014
Lead optimization of 1,4-azaindoles as antimycobacterial agents.
Journal: Journal of medicinal chemistry
Published: May 31, 2014
4-aminoquinolone piperidine amides: noncovalent inhibitors of DprE1 with long residence time and potent antimycobacterial activity.
Journal: Journal of medicinal chemistry
Published: May 30, 2014
Novel N-linked aminopiperidine-based gyrase inhibitors with improved hERG and in vivo efficacy against Mycobacterium tuberculosis.
Journal: Journal of medicinal chemistry
Published: May 09, 2014
Benzimidazoles: novel mycobacterial gyrase inhibitors from scaffold morphing.
Journal: ACS medicinal chemistry letters
Published: April 29, 2014
Last Updated: 09/26/2026