Randomised, Open-label and Parallel Group Trial to Investigate the Effects of Oral BI 685509 Alone or in Combination With Empagliflozin on Portal Hypertension After 8 Weeks Treatment in Patients With Clinically Significant Portal Hypertension (CSPH) in Compensated Cirrhosis

Status: Terminated
Location: See all (31) locations...
Intervention Type: Drug
Study Type: Interventional
Study Phase: Phase 2
SUMMARY

This study is open to adults with liver cirrhosis caused by hepatitis B, hepatitis C or nonalcoholic steatohepatitis (NASH). People can join this study if they have high blood pressure in the portal vein (main vessel going to the liver). The purpose of this study is to find out whether a medicine called Avenciguat (BI 685509) taken alone or in combination with a medicine called empagliflozin helps people with this condition. Participants take Avenciguat (BI 685509) as tablets twice a day for 8 weeks. Half of the participants with NASH who also have type 2 diabetes take empagliflozin as tablets once a day in addition to Avenciguat (BI 685509). Participants are in the study for about 3 months. During this time, they visit the study site about 10 times. At 2 of the visits, the doctors check the pressure in a liver vein to see whether the treatment works. This is done with a catheter (a long thin tube) and gives information about the pressure in the portal vein. The doctors also regularly check participants' health and take note of any unwanted effects.

Eligibility
Participation Requirements
Sex: All
Minimum Age: 18
Maximum Age: 75
Healthy Volunteers: f
View:

• Signed and dated written informed consent in accordance with ICH-GCP and local legislation prior to admission to the trial

• Male or female who is ≥ 18 (or who is of legal age in countries where that is greater than 18) and ≤ 75 years old at screening (Visit 1a)

• Clinical signs of Clinically Significant Portal Hypertension (CSPH) as described by either one of the points below. Each trial patient must have a gastroscopy during the screening period (Visit 1b) or within 6 months prior to screening (Visit 1b).

‣ documented endoscopic proof of oesophageal varices and / or gastric varices at screening (Visit 1b) or within 6 months prior to screening (Visit 1b)

⁃ documented endoscopic-treated oesophageal varices as preventative treatment

• CSPH defined as baseline Hepatic Venous Pressure Gradient (HVPG) ≥ 10 mmHg (measured at Visit 1c), based on a local interpretation of the pressure tracing

• Diagnosis of compensated cirrhosis due to Hepatitis C virus (HCV), Hepatitis B virus (HBV), or Non-Alcoholic Steatohepatitis (NASH) with or without Type 2 Diabetes Melitus (T2DM). Diagnosis of cirrhosis must be based on histology (historical data is acceptable) or on clinical evidence of cirrhosis (e.g. platelet count \< 150 x 109/L \[150 x 103/microlitre (μL)\], nodular liver surface on imaging or splenomegaly etc.) Diagnosis of NASH based on either i. Current or historic histological diagnosis of NASH OR steatosis OR ii. Clinical diagnosis of NASH based on historic or current imaging diagnosis of fatty liver (Fibroscan, Ultrasound (US), Magnetic Resonance Imaging (MRI), Computed Tomography (CT)) AND at least 2 current or historic comorbidities of the metabolic syndrome (overweight/obesity, T2DM, hypertension, hyperlipidemia)

• Willing and able to undergo HVPG measurements per protocol (based on Investigator judgement)

• If receiving statins must be on a stable dose for at least 3 months prior to screening (Visit 1b), with no planned dose change throughout the trial

• If receiving treatment with Non-Selective Beta-Blocker (NSBBs) or carvedilol must be on a stable dose for at least 1 months prior to screening (Visit 1b), with no planned dose change throughout the trial

• Further inclusion criteria apply

Locations
United States
California
California Liver Research Institute
Pasadena
Inland Empire Clinical Trials, LLC
Rialto
Florida
Floridian Clinical Research-Miami Lakes-68368
Miami Lakes
Texas
American Research Corporation
San Antonio
Other Locations
Argentina
Hospital Britanico de Buenos Aires
Caba
Hospital Italiano de Buenos Aires
Caba
Austria
AKH - Medical University of Vienna
Vienna
Belgium
Edegem - UNIV UZ Antwerpen
Edegem
Canada
Centre Hospitalier de l'Universite de Montreal (CHUM)
Montreal
China
Beijing Friendship Hospital
Beijing
NanFang Hosptial
Guangzhou
The Affiliated Hospital of Hangzhou Normal University
Hangzhou
Zhongshan Hospital Affiliated to Fudan University
Shanghai
Denmark
Hvidovre Hospital
Hvidovre
France
HOP Beaujon
Clichy
HOP Rangueil
Toulouse
Germany
Medizinische Hochschule Hannover
Hanover
Universitätsmedizin der Johannes Gutenberg-Universität Mainz
Mainz
Universitätsklinikum Münster
Münster
Israel
Rambam Medical Center
Haifa
Western Galilee Hospital
Nahariya
Italy
Ospedale Civile di Baggiovara
Baggiovara (mo)
Azienda Ospedaliera Policlinico di Modena
Modena
Policlinico Paolo Giaccone
Palermo
Japan
National Hospital Organization Yokohama Medical Center
Kanagawa, Yokohama
Osaka Metropolitan University Hospital
Osaka, Osaka
Netherlands
Amsterdam UMC, location VUMC
Amsterdam
Romania
Regional Institute of Gastroenterology Hepatology Prof. Dr. O. Fodor
Cluj-napoca
Singapore
Singapore General Hospital
Singapore
Spain
Hospital Vall d'Hebron
Barcelona
Hospital Ramón y Cajal
Madrid
Time Frame
Start Date: 2022-06-28
Completion Date: 2024-06-07
Participants
Target number of participants: 90
Treatments
Experimental: Patients with HBV - avenciguat
Patients with Hepatitis B Virus (HBV) were administered one film-coated tablet of avenciguat orally twice a day. The two doses were ideally taken at least 10 hours apart. The starting dose was 1 milligram (mg), which, if tolerated, was up-titrated to 2 mg one week later. If this dose was also tolerated, a second up-titration to 3 mg occured after another week. Patients remained on the highest dose for the remainder of the treatment period, until 8 weeks of treatment.
Experimental: Patients with HCV - avenciguat
Patients with Hepatitis C Virus (HCV) were administered one film-coated tablet of avenciguat orally twice a day. The two doses were ideally taken at least 10 hours apart. The starting dose was 1 milligram (mg), which, if tolerated, was up-titrated to 2 mg one week later. If this dose was also tolerated, a second up-titration to 3 mg occured after another week. Patients remained on the highest dose for the remainder of the treatment period, until 8 weeks of treatment.
Experimental: Patients with NASH with or without T2DM - avenciguat
Patients with Non-Alcoholic Steatohepatitis (NASH) with or without type 2 Diabetes Mellitus (T2DM) were administered one film-coated tablet of avenciguat orally twice a day. The two doses were ideally taken at least 10 hours apart. The starting dose was 1 milligram (mg), which, if tolerated, was up-titrated to 2 mg one week later. If this dose was also tolerated, a second up-titration to 3 mg occured after another week. Patients remained on the highest dose for the remainder of the treatment period, until 8 weeks of treatment.
Experimental: Patients with NASH with T2DM - avenciguat + empagliflozin
Patients with Non-Alcoholic Steatohepatitis (NASH) with type 2 Diabetes Mellitus (T2DM) were administered one film-coated tablet of avenciguat orally twice a day. The two doses were ideally taken at least 10 hours apart. The starting dose was 1 milligram (mg), which, if tolerated, was up-titrated to 2 mg one week later. If this dose was also tolerated, a second up-titration to 3 mg occured after another week. Patients remained on the highest dose for the remainder of the treatment period, until 8 weeks of treatment.~Patients were additionally administered one 10 mg film-coated tablet of empagliflozin orally once a day.
Sponsors
Leads: Boehringer Ingelheim

This content was sourced from clinicaltrials.gov